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Discovery of a Highly Selective Sigma-2 Receptor Ligand, 1-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-3-methyl-1H-benzo[d]imidazol-2(3H)-one (CM398), with Drug-Like Properties and Antinociceptive Effects In Vivo

Sebastiano Intagliata; Abhisheak Sharma; Tamara I. King; Christophe Mesangeau; Michael Seminerio; Frederick T. Chin; Lisa L. Wilson; Rae R. Matsumoto; Jay P. McLaughlin; Bonnie A. Avery; Christopher R. McCurdy
The AAPS Journal · Vol. 22, Issue 5 · 2020

Abstract

Abstract is unavailable.

Bibliographic Information

JournalThe AAPS Journal
PublisherSpringer
Publication Date2020-09-01
Publication Year2020
Volume22
Issue5
Document TypeJournal Article
eISSN1550-7416
DOI10.1208/s12248-020-00472-x

Access Information

NARA Access Coverage1999-01-01~Current
Journal Homepagehttps://www.springer.com/journal/12248
Publisher PageOpen Publisher Page
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