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Identification of reversible OATP1B1 and time-dependent CYP3A4 inhibition as the major risk factors for drug-induced cholestasis (DIC)

Vlasia Kastrinou-Lampou; Raquel Rodríguez-Pérez; Birk Poller; Felix Huth; Zsuzsanna Gáborik; Beáta Mártonné-Tóth; Csilla Temesszentandrási-Ambrus; Heiko S. Schadt; Gerd A. Kullak-Ublick; Michael Arand; Gian Camenisch
Archives of Toxicology · Vol. 98, Issue 10 · pp. 3409-3424 · 2024

Abstract

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Bibliographic Information

JournalArchives of Toxicology
PublisherSpringer
Publication Date2024-10-01
Publication Year2024
Volume98
Issue10
Pages3409-3424
Document TypeJournal Article
Print ISSN0340-5761
eISSN1432-0738
DOI10.1007/s00204-024-03794-3

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NARA Access Coverage1930-01-01~Current
Journal Homepagehttps://www.springer.com/journal/204
Publisher PageOpen Publisher Page
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