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Physiologically based pharmacokinetic combined BTK occupancy modeling for optimal dosing regimen prediction of acalabrutinib in patients alone, with different CYP3A4 variants, co-administered with CYP3A4 modulators and with hepatic impairment

Lifang Xu; Shuang Yu; Huining Liu; Bowen Yi; Guopeng Wang; Yang Liu
European Journal of Clinical Pharmacology · Vol. 78, Issue 9 · pp. 1435-1446 · 2022

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Bibliographic Information

JournalEuropean Journal of Clinical Pharmacology
PublisherSpringer
Publication Date2022-09-01
Publication Year2022
Volume78
Issue9
Pages1435-1446
Document TypeJournal Article
Print ISSN0031-6970
eISSN1432-1041
DOI10.1007/s00228-022-03338-7

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NARA Access Coverage1968-01-01~Current
Journal Homepagehttps://www.springer.com/journal/228
Publisher PageOpen Publisher Page
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